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½üÆÚ´ú±íÐÔSCIÂÛÎÄ£º1. Renren Bai, Zhen Wei, Jie Liu, Weijia Xie, Hequan Yao, Xiaoming Wu*, Jieyun Jiang, Qiujuan Wang, Jinyi Xu*. Synthesis and biological evaluation of 4¡ä-[(benzimidazole-1-yl)methyl]biphenyl-2-sulfonamide derivatives as dual angiotensin II/endothelin A receptor antagonists. Bioorganic & Medicinal Chemistry, 2012, 20(15), 4661-4667.2. Dahong Li, Hao Cai, Bowen Jiang, Guyue Liu, Yuetong Wang, Lei Wang, Hequan Yao, Xiaoming Wu*, Yijun Sun, Jinyi Xu*. Synthesis of spirolactone-type diterpenoid derivatives from kaurene-type oridonin with improved antiproliferative effects and their apoptosis-inducing activity in human hepatoma Bel-7402 cells. European Journal of Medicinal Chemistry, 2013, 59, 322-328.3. Ziyuan Li, Ling Ma, JinyiXu, Lingyi Kong, Xiaoming Wu*, Hequan Yao*. Pd(II)-catalyzed direct C5-arylation of azole-4-carboxylates through double C-H bond cleavage. Chemical Communications, 2012, 48(31), 3763-3765.4. Lei Zhao, Ziyuan Li, Lin Chang, JinyiXu, Hequan Yao*, Xiaoming Wu*. Efficient Construction of Fused Indolines with a 2-Quaternary Center via an Intramolecular Heck Reaction with a Low Catalyst Loading. Organic Letters, 2012, 68(14), 2066-2069.5. Renren Bai, Xue Yang, Wen Hong, Yiqun Tang, Shengtao Xu, Hequan Yao, Jieyun Jiang, Jie Liu, Mingqin Shen, Xiaoming Wu*, Jinyi Xu*. Novel hybrids of natural isochroman-4-one bearing N-substituted isopropanolamine as potential antihypertensive candidates. Bioorganic & Medicinal Chemistry, 2013, 21, 2495-2502.6. Dan Liu, Weijia Xie*, Long Liu, Hequan Yao, Jinyi Xu, Genzoh Tanabe, Osamu Muraoka, Xiaoming Wu*. Synthetic study on neoponkoranol and its side chain epimer as potent a-glucosidase inhibitors, optimization of protecting group. Tetrahedron Letters. 2013, 54, 6333-6336.7. Dahong Li, Shengtao Xu, Hao Cai, Lingling Pei, Lei Wang, Hequan Yao, Xiaoming Wu*, Jieyun Jiang, Yijun Sun, Jinyi Xu*. Library construction and biological evaluation of novel enmein-type diterpenoid analogs as potential anticancer agents. Chem. Med. Chem., 2013, 8: 812-818.8. Dahong Li, Shengtao Xu, Hao Cai, Lingling Pei, Hengyuan Zhang, Lei Wang, Hequan Yao, Xiaoming Wu*, Jieyun Jiang, Yijun Sun, Jinyi Xu*. Enmein-type diterpenoid analogs from natural kaurene-type oridonin: synthesis and their antitumor biological evaluation Eur. J. Med. Chem. 2013, 64, 215-221.9. Long Liu, Chengqian Wang, Dan Liu, Weigang He, Jinyi Xu, Aijun Lin, Hequan Yao, Genzoh Tanabe, Osamu Muraoka, Weijia Xie,* Xiaoming Wu,* Construction of 3,6-Anhydrohexosides via Intramolecular Cyclization of Triflates and Its Application to the Synthesis of Natural Product Isolated from Leaves of Sauropus rostratus. Organic Letters 2014, 16, 5004-5007.10. Bo Jiang, Xiaojing Huang, Hequan Yao, Jieyun Jiang, Xiaoming Wu*, Siyi Jiang, Qiujuan Wang, Tao Lu and Jinyi Xu*. Discovery of potential anti-inflammatory drugs: diaryl-1,2,4-triazoles bearing N-hydroxyurea moiety as dual inhibitors of cyclooxygenase-2 and 5-lipoxygenase. Org. Biomol. Chem., 2014, 12, 2114-2127.