ÍõТΰ:¸±½ÌÊÚ£¬Ë¶Ê¿Éúµ¼Ê¦¡£
µç»°£º(010)-82805203
E-mail: xiaoweiwang@bjmu.edu.cn
ͨѶµØÖ·£º±±¾©Êк£µíÇøÑ§ÔºÂ·38ºÅ±±¾©´óѧҩѧԺ Óʱࣺ100191
1988Äê±ÏÒµÓÚ±±¾©Ò½¿Æ´óѧҩѧԺ£¬Í¬ÄêÁôУ´ÓÊÂÓлú»¯Ñ§µÄ½ÌѧÓë¿ÆÑй¤×÷¡£ÀúÈα±¾©´óѧҩѧԺÖú½Ì¡¢½²Ê¦¡¢¸±½ÌÊÚ¡£2008ÄêÔÚÈÕ±¾½øÐÞ¡£ÔÚ´ËÆÚ¼ä£¬²ÎÓëÁ˶àÏî¿ÎÌâµÄÑо¿£¬ÆäÖаüÀ¨Óë±±¾©ÊпÆÎ¯ÏÂÊôÑо¿ËùºÏ×÷µÄ×Ïɼ´¼µÄ°ëºÏ³É£»ÌÇÜÕøÒÖÖÆ¼ÁÒÔ¼°Ñª¹Ü½ôÕÅËØIIÊÜÌåÞ׿¹¼ÁµÄ»îÐԲⶨ¡£2000ÄêÆð£¬Ò»Ö±´ÓÊ¿¹°¬×̲¡Ò©ÎïµÄÑо¿¹¤×÷£¬³Ðµ£ºÍ²ÎÓë¿Æ¼¼²¿¡°Ê®Ò»ÎåÖ§³Å¼Æ»®¡±¡¢¹ú¼Ò×ÔÈ»¿ÆÑ§»ù½ð¡¢±±´ó·½Õý»ù½ðµÈÏîÄ¿¡£¶ÔHIV²¡¶¾×÷ÓÃµÄ°Ðµã½øÐÐÁËÏ꾡Ñо¿£¬ÌرðÊÇÔÚ¶ÔÄæ×ªÂ¼Ã¸ÒÖÖÆ¼ÁµÄ×÷ÓûúÀí¡¢¹¹Ïó¹ØÏµ¼°ÄÍÒ©ÎÊÌâÑо¿µÄͬʱ£¬½áºÏ¼ÆËã»ú¸¨ÖúÉè¼Æ£¬ºÏ³ÉÁË6ÖÖÀàÐͽü300¶à¸ö»¯ºÏÎÆäÖÐÒ»¸ö»¯ºÏÎïÒѾ½øÈëÁËÁÙ´²Ç°µÄÑо¿¡£²¢ÉêÇëÁ˶àÏîרÀû¡£½üÆÚÓÖ¿ªÕ¹ÁË¿¹HIVË«°ÐµãÒ©ÎïµÄÑо¿¡£ÓÉÓÚһЩ»¯ºÏÎïÉè¼ÆÀíÄîÐÂÓ±£¬¶øµÃµ½Á˹úÍâר¼ÒµÄºÃÆÀ£¬ÔÚ¹úÄÚÍâ·¢±íÁË¶àÆªÆÚ¿¯ÂÛÎļ°ÖØ´ó»áÒéÂÛÎÄ¡£
Ö÷ÒªÑо¿·½Ïò£º
¶ÔHIV²¡¶¾×÷ÓÃµÄ°Ðµã£¬ÌØ±ð¶ÔÄæ×ªÂ¼Ã¸ÒÖÖÆ¼ÁµÄ×÷ÓûúÀí¡¢¹¹Ïó¹ØÏµ¼°ÄÍ
Ò©ÎÊÌâ½øÐÐÑо¿¡£½áºÏ¼ÆËã»ú¸¨ÖúÒ©ÎïÉè¼Æ¡¢·Ö×ÓÄ£ÄâµÈ¼¼Êõ£¬Éè¼Æ¶àÖÖÀàÐ͵ĵ¥°Ðµã¼°¶à°ÐµãÒÖÖÆ¼Á£¬Ï£Íû´ÓÖÐÕÒµ½¸÷ÏîÐÔÄܸüΪÓÅÁ¼µÄ¿¹ÄÍÒ©ÐԵĿ¹HIV²¡¶¾Ïȵ¼»¯ºÏÎï¡£
1. ¿¹HIV-1Äæ×ªÂ¼Ã¸(RT)µ¥°ÐµãÒÖÖÆ¼ÁµÄÉè¼ÆºÏ³É¼°»îÐÔÆÀ¹À¡£
2. ¿¹HIV²¡¶¾Äæ×ªÂ¼£¨RT£©/ÕûºÏø(IN)Ë«°ÐµãÒÖÖÆ¼ÁµÄÉè¼ÆºÏ³É¼°»îÐÔÆÀ¹À
3. ¿¹HIV²¡¶¾Äæ×ªÂ¼£¨RT£©/½øÈë(EN)Ë«°ÐµãÒÖÖÆ¼ÁµÄÉè¼ÆºÏ³É¼°»îÐÔÆÀ¹À
½üÄê²ÎÓë¼°Ö÷³ÖµÄ¿ÆÑÐÏîÄ¿£º
1. ¹ú¼Ò×ÔÈ»¿ÆÑ§»ù½ð¡°»·¸ýæéà×à¤ÀàÐÂÐͷǺËÜÕ¿¹°¬×̲¡Ò©ÎïµÄÉè¼ÆºÏ³É¼°»îÐÔÑо¿¡±
2. ²©Ê¿µã»ù½ð¡°»·¸ü²¢à×à¤ÀàÐÂÐͷǺËÜÕ¿¹°¬×̲¡Ò©ÎïµÄÉè¼ÆºÏ³ÉºÍ»îÐÔÑо¿¡±
3. ¹ú¼Ò×ÔÈ»¿ÆÑ§»ù½ð¡°»ùÓÚDAPY/S-DABO½á¹¹µÄÐÂÐͷǺËÜÕÀàÄæ×ªÂ¼Ã¸ÒÖÖÆ¼ÁµÄÑо¿¡±
4. ±±¾©´óѧ×ÛºÏÐÔ´´ÐÂÒ©ÎïÑо¿¼¼Êõ´óƽ̨ÐÂÒ©Æ·ÖÖ¡°à×à¤ÍªÀ࿹HIVÒ©ÎïµÄÁÙ´²Ç°Ñо¿¡±
5. ±±´ó·½Õý´´ÐÂÒ©ÎïÑо¿»ù½ð¡°¿¹HIVÒ©ÎïµÄÑз¢¡±
´ú±íÐÔÂÛÎÄ£º
1.Xiaowei Wang, Qinghua Lou, Ying Guo, Yang Xu, Zhili Zhang and Junyi Liu£¬The design and synthesis of 9-phenylcyclohepta[d] pyrimidine-2, 4-dione derivatives as potent non- nucleoside inhibitors of HIV reverse transcriptase. Organic & Biomolecular Chemistry 2006, 4, 3252¨C3258
2.Inhibitory activity of 9-phenylcyclohepta[d]pyrimidinedione derivatives against different strains of HIV-1 as non-nucleoside reverse transcriptase inhibitors. Virology Journal 2011, 8:230 (accepted)
3. Xiaowei Wang , Yanli Chen ; Ying Guo ; Amin Li ; Xiaoyan Mab; Junyi Liu, Synthesis of 1-(Alkyl)-5-Dimethylamino-6- Phenethyluracils as Potent Non- nucleoside HIV-1 RT Inhibitors Synthetic Communications 37: 2421¨C2431, 2007
4. Libo Gao ; Shigan Fu; Hui Li; Xiaowei Wang; Junyi Liu ;Han Liu; Liyuan Guo; Xinhua Liu; Mengsen Li; Michael A. McNutt; Gang Li, Pyrimidone derivative inhibits simian immunodeficiency virus-induced apoptosis of CEM x174 cells, Cell Biology International 33 (2009) 207-216
5. Xiao Lu, Yanli Chen, Ying Guo, Zhenming Liu, Yawei Shi, Yang Xu, Xiaowei Wang and Junyi Liu, The Design and Synthesis of N-1 alkylated 5-aminoaryalkyl substituted 6-methyluracils as potential non-nucleoside HIV-1 RT Inhibitors Bioorganic Medicinal Chemistry 15 (2007) 7399¨C7407
6. Hua Qin, Jianfang Zhang, Chang Liu, Ying Guo, Siwei Zhang, Zhili Zhang, Xiaowei Wang, Liangren Zhang, Junyi Liu, Synthesis and biological evaluation of novel 2-arylalkylthio-4-amino-6-benzyl pyrimidines as potent HIV-1 non-nucleoside reverse transcriptase inhibitors, Bioorganic Medicinal Chemistry Letter 2009.04.051
7. Hua Qin, Chang Liu, Ying Guo, Ruiping Wang, Jianfang Zhang, Liying Ma, Zhili Zhang, Xiaowei Wang, Yuxin Cui, Junyi Liu. Synthesis and biological evaluation of novel C5 halogen-functionalized S-DABO as potent HIV-1 non-nucleoside reverse transcriptase inhibitors. Bioorganic & Medicinal Chemistry 2010, 18: 3231¨C3237.
8.Xiaowei Wang, Yu Gao, Yang Xu, Li Li, Zhili Zhang, Junyi Liu. An efficient preparation of a photolabile agent MNI-glu by regioselective nitration of 4-methoxyindoline derivative. Synthetic Communications 2009, 39(22); 4030-4038
9.Li A-min, Wang Xiao-wei, Zhang Zhi-li, Cheng Zhi-jian and Liu Jun-yi. Regioselective Deprotection of 1,3-Dibenzyl-5-(N,N-dimethylamino)-6-phenylethyluracil. Chemical Research, Chinese University. 2008, 24(6): 1-4
ÉêÇë·¢Ã÷רÀû£º
201010208308.7ÐÂÐÍHEPTÀàHIV-1Äæ×ªÂ¼Ã¸ÒÖÖÆ¼ÁµÄÖÆ±¸¼°ÆäÓ¦ÓÃ
201010136763.0 6-Üлù-1-ÒÒÑõ¼×»ù-5-Òì±û»ùëåà×à¤(Emivirine)¼°ÆäÀàËÆÎïµÄкϳɷ½·¨
201010515280.1 ÐÂÐÍßÁà¤ÍªÀàHIV-1Äæ×ªÂ¼Ã¸ÒÖÖÆ¼ÁµÄÖÆ±¸¼°ÆäÓ¦ÓÃ
±±¾©´óѧҩѧԺ»¯Ñ§ÉúÎïѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØË¶Ê¿Ñо¿Éúµ¼Ê¦ÐÅÏ¢£ºÍõТΰ
±¾Õ¾Ð¡±à Ãâ·ÑöλÔÓéÀÖ¹Ù·½appÏÂÔØÍø/2016-06-22
Ïà¹Ø»°Ìâ/Ò©Îï Éè¼Æ ²¡¶¾ »ù½ð ±±¾©´óѧ
±±¾©´óѧҩѧԺ˶ʿÑо¿Éúµ¼Ê¦ÐÅÏ¢
±±¾©´óѧҩѧԺҩÎﻯѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØË¶Ê¿Ñо¿Éúµ¼Ê¦ÐÅÏ¢Òѹ«²¼£¬ÏêÇéÈçÏ£º öλÔÓéÀֵǼÈë¿ÚÏÂÔØ µ¼Ê¦ÐÕÃû Ñо¿·½Ïò ...µ¼Ê¦ÐÅÏ¢ ±¾Õ¾Ð¡±à Ãâ·ÑöλÔÓéÀÖ¹Ù·½appÏÂÔØÍø 2016-06-22±±¾©´óѧҩѧԺҩÎﻯѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØË¶Ê¿Ñо¿Éúµ¼Ê¦ÐÅÏ¢£ºÌÀо°
Dr. Xinjing TangState Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences,Peking UniversityTel: +86 10 82805635E-mail: x ...µ¼Ê¦ÐÅÏ¢ ±¾Õ¾Ð¡±à Ãâ·ÑöλÔÓéÀÖ¹Ù·½appÏÂÔØÍø 2016-06-22±±¾©´óѧҩѧԺҩÎﻯѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØË¶Ê¿Ñо¿Éúµ¼Ê¦ÐÅÏ¢£ºÍõ³¬
Íõ ³¬ ½ÌÊÚ Àíѧ²©Ê¿ °ì¹«µç»°£º010-82805049 µç×ÓÐÅÏ䣺chaowang@bjmu.edu.cnÑо¿·½Ïò£ºÒ©Îﻯѧ£¬¶àëÄ»¯Ñ§1961Äê4Ô³öÉú¡£1995ÄêÓÚ±±¾©Ò½¿Æ´óѧҩѧԺ»ñÀíѧ²©Ê¿Ñ§Î»¡£2003Äê½úÉýΪ½ÌÊÚ¡£Ë¶Ê¿Éúµ¼Ê¦¡£2001¡¢£2002ÄêÔÚ·¨¹ú¹ú¼Ò¿ÆÑÐÖÐÐĵÄ"½á¹¹ÉúÎïѧÑо¿Ëù" ...µ¼Ê¦ÐÅÏ¢ ±¾Õ¾Ð¡±à Ãâ·ÑöλÔÓéÀÖ¹Ù·½appÏÂÔØÍø 2016-06-22±±¾©´óѧҩѧԺҩÎﻯѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØË¶Ê¿Ñо¿Éúµ¼Ê¦ÐÅÏ¢£ºÁõÕñÃ÷
ÁõÕñÃ÷Àíѧ²©Ê¿£¬¸±Ñо¿Ô±Ò©Îﻯѧ£¬Ò©ÎïÉè¼Æµç»° & ´«Õæ: +86-10-82805514 +86-10-82802724ÁªÏµÓÊÏä: zmliu@bjmu.edu.cnѧϰ¾Àú:1996-2000 Àíѧѧʿ£¬±±¾©Ò½¿Æ´óѧҩѧԺҩÎﻯѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØ2000-2005 Àíѧ²©Ê¿£¬±±¾©´óѧ»¯Ñ§Óë·Ö×Ó¹¤³ÌѧԺÎïÀí ...µ¼Ê¦ÐÅÏ¢ ±¾Õ¾Ð¡±à Ãâ·ÑöλÔÓéÀÖ¹Ù·½appÏÂÔØÍø 2016-06-22±±¾©´óѧҩѧԺҩ¼ÁѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØË¶Ê¿Ñо¿Éúµ¼Ê¦ÐÅÏ¢£º·¶ÌïÔ°
·¶ÌïÔ° ²©Ê¿ ¸±½ÌÊڵ绰/´«Õ棺82801584£¬ÓÊÏ䣺tianyuan_fan@bjmu.edu.cn×Ô1983ÄêÔÚ±±¾©´óѧҩѧԺѧϰºÍ¹¤×÷£¬ÆÚ¼äÂ½Ðø»ñµÃѧʿ£¨1988Ä꣩¡¢Ë¶Ê¿£¨1991Ä꣩ºÍ²©Ê¿£¨2001Ä꣩ѧλ£¬Ôø·Ö±ðµ½Ïã¸ÛÖÐÎÄ´óѧ£¨1996Ä꣩ºÍÈÕ±¾ÐÇÒ©¿Æ´óѧ£¨2002Ä꣩·ÃÎÊѧϰ¡£´ÓÊÂÒ© ...µ¼Ê¦ÐÅÏ¢ ±¾Õ¾Ð¡±à Ãâ·ÑöλÔÓéÀÖ¹Ù·½appÏÂÔØÍø 2016-06-22±±¾©´óѧҩѧԺҩ¼ÁѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØË¶Ê¿Ñо¿Éúµ¼Ê¦ÐÅÏ¢£ºÁõÑÞ
Áõ ÑÞ ¸±½ÌÊÚ, ˶ʿÉúµ¼Ê¦±±¾©´óѧҩѧԺҩ¼Áѧϵ¸±Ö÷Èα±¾©Êк£µíÇøÑ§ÔºÂ·38ºÅ£¬Óʱà 100191Tel: (+8610) 82801508Email: yanliu@bjmu.edu.cn1986ÄêÔÚɽ¶«´óѧ»¯Ñ§Ïµ»ñµÃÀíѧѧʿѧλ¡£1989ÄêÔÚɽ¶«´óѧ»¯Ñ§Ïµ»ñµÃÀíѧ˶ʿѧλ¡£Í¬Äê8Ôµ½±±¾©Ò½¿Æ´ó ...µ¼Ê¦ÐÅÏ¢ ±¾Õ¾Ð¡±à Ãâ·ÑöλÔÓéÀÖ¹Ù·½appÏÂÔØÍø 2016-06-22±±¾©´óѧҩѧԺҩ¼ÁѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØË¶Ê¿Ñо¿Éúµ¼Ê¦ÐÅÏ¢£ºÍõ¼á³É
Íõ¼á³É ¸±½ÌÊÚ¡¢Ë¶Ê¿Éúµ¼Ê¦Asso. Prof. Jian-Cheng WangTel & Fax : (010) 8280 2683 (Office)£»8280 5764 (Lab) Email: wang-jc@bjmu.edu.cn1992Äê9Ô¡ª1997Äê7Ô ±±¾©Ò½¿Æ´óѧ ҩѧԺӦÓû¯Ñ§×¨ ...µ¼Ê¦ÐÅÏ¢ ±¾Õ¾Ð¡±à Ãâ·ÑöλÔÓéÀÖ¹Ù·½appÏÂÔØÍø 2016-06-22±±¾©´óѧҩѧԺҩ¼ÁѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØË¶Ê¿Ñо¿Éúµ¼Ê¦ÐÅÏ¢£ºÍõѧÇå
ÍõѧÇå ²©Ê¿£¬¸±½ÌÊÚ£¬Ë¶Ê¿Ñо¿Éúµ¼Ê¦µç»°£º010-82801584,µç×ÓÐÅÏ䣺wangxq@bjmu.edu.cn1989.9-1993.7 ±±¾©Ò½¿Æ´óѧҩѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØÑ§Ï°£¬»ñѧʿѧλ¡£2001.9-2003.7ÄêÓÚ±±¾©´óѧҩ¼ÁѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØÔÚְѧϰ£¬»ñ˶ʿѧλ¡£2005.9-2008.7ÄêÓÚÖйú¿ÆÑ§ÔºÉúÎïÎïÀíÑÐ ...µ¼Ê¦ÐÅÏ¢ ±¾Õ¾Ð¡±à Ãâ·ÑöλÔÓéÀÖ¹Ù·½appÏÂÔØÍø 2016-06-22±±¾©´óѧҩѧԺҩ¼ÁѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØË¶Ê¿Ñо¿Éúµ¼Ê¦ÐÅÏ¢£ºÖÜÌïÑå
ÖÜÌïÑ岩ʿ¸±½ÌÊÚ˶ʿÉúµ¼Ê¦µç»°/´«Õ棺(10)-82801717µç×ÓÐÅÏ䣺tianyanzhou@bjmu.edu.cn¼òÀú·Ö±ðÓÚ1992 Äê¡¢1998 ÄêÔÚ±±¾©Ò½¿Æ´óѧҩѧԺ»ñµÃѧʿºÍ˶ʿѧ룬98ÄêÁôУÖÁ½ñÒ»Ö±ÔÚ±±¾©´óѧҩѧԺҩ¼Á½ÌÑÐÊÒ¹¤×÷£¬²¢ÓÚ2006 ÄêÈ¡µÃÒ©¼Áѧ²©Ê¿Ñ§Î»¡£Ôøµ½Ïã¸ÛÀí¹¤´óѧ£¨ ...µ¼Ê¦ÐÅÏ¢ ±¾Õ¾Ð¡±à Ãâ·ÑöλÔÓéÀÖ¹Ù·½appÏÂÔØÍø 2016-06-22±±¾©´óѧҩѧԺÉúҩѧöλÔÓéÀֵǼÈë¿ÚÏÂÔØË¶Ê¿Ñо¿Éúµ¼Ê¦ÐÅÏ¢£º³µÇìÃ÷
³µÇìÃ÷ ҩѧ²©Ê¿ ½ÌÊÚ ½ÌÊÚ¹ú¼Ò½Ü³öÇàÄê»ù½ð»ñµÃÕßÑо¿ÁìÓò£ºÖÐÒ©»¯Ñ§¼°Ò©Îï´úлµç»°/´«Õ棺+86-10-82802468 ÁªÏµÓÊÏ䣺cheqingming2008@sina.com¸öÈ˼òÀú96.06--ÖÁ½ñ ±±¾©´óѧҩѧԺÖÐÒ©Ñо¿ÊÒ½ÌÊÚÑо¿·½Ïò (1)ÖÐÒ©ÓÐЧ³É·ÖµÄ»¯Ñ§Ñо¿ (2)ÖÐÒ©³É·ÖµÄѪÇåÒ©Îï ...µ¼Ê¦ÐÅÏ¢ ±¾Õ¾Ð¡±à Ãâ·ÑöλÔÓéÀÖ¹Ù·½appÏÂÔØÍø 2016-06-22
